Available PET Radioligands for Human Use

List of available PET radioligands injected into humans

 

Target

 

Radiotracer

 

Benzodiazepine antagonist

 

[11C]Flumazenil

 

Cannabinoid receptor type 1

 

[11C]JHU75528

 

Cerebral blood flow

 

[15O]water

 

Dopamine D2/D3 receptor

 

[11C]PHNO

 

Dopamine D2/D3 receptor

 

[11C]Raclopride

 

Dopamine transporter

 

[11C]PE2I

 

Extrastriatal dopamine D2

 

[11C]FLB457

 

Fibrillar amyloid-beta (Aβ) plaques

 

[11C]PIB

 

Fibrillar amyloid-beta (Aβ) plaques

 

[18F]BPIB

 

Glucose metabolism

 

[18F]FDG

 

Glycine transporter 1

 

[18F]CFpyPB

 

Histamine-3

 

[11C]GSK189254

 

Hypoxia

 

[18F]FMISO

 

Kappa antagonist

 

[11C]LY2795050

 

Kappa opioid

 

[11C]GR103545

 

Metabotropic glutamate receptor 5

 

[11C]ABP688

 

Metabotropic glutamate receptor 5

 

[18F]FPEB

 

Myocardial blood flow

 

82Rb

 

Nicotinic a4b2 receptors

 

[18F]NCFHEB

 

Norepinephrine transporter

 

[11C]MRB

 

Peripheral benzodiazepine receptor

 

[11C]PBR28

 

Phosphodiesterase-2A

 

[18F]PF-05270430

 

Serotonin 5HT1B receptor

 

[11C]P943

 

Serotonin 5-HT1A receptor antagonist

 

[11C]CUMI

 

Serotonin 5-HT2A receptor

 

[11C]MDL100907

 

Serotonin 5HT4 receptor

 

[11C]SB-207145

 

Serotonin 5-HT6 receptor

 

[11C]GSK-215083

 

Serotonin Transporter

 

[11C]AFM

 

Serotonin Transporter

 

[11C]DASB

 

Vesicular monoamine transporter 2

 

[18F](+)FP-DTBZ

 

Tracking protein synthesis

 

[11C]Methionine

Gallery of selected PET Radioligands