2018
Curcumin Acts as a Positive Allosteric Modulator of α 7-Nicotinic Acetylcholine Receptors and Reverses Nociception in Mouse Models of Inflammatory Pain
El Nebrisi E, Bagdas D, Toma W, Al Samri H, Brodzik A, Alkhlaif Y, Yang K, Howarth F, Damaj I, Oz M. Curcumin Acts as a Positive Allosteric Modulator of α 7-Nicotinic Acetylcholine Receptors and Reverses Nociception in Mouse Models of Inflammatory Pain. Journal Of Pharmacology And Experimental Therapeutics 2018, 365: 190-200. PMID: 29339457, PMCID: PMC7947331, DOI: 10.1124/jpet.117.245068.Peer-Reviewed Original ResearchConceptsEffect of curcuminPositive allosteric modulatorsMouse modelVisceral painAntinociceptive effectNACh receptorsAcetylcholine receptorsAllosteric modulatorsΑ7 nicotinic acetylcholine receptorVisceral pain modelHuman nicotinic acetylcholine receptorNicotinic acetylcholine receptorsInflammatory painPain modelNociceptive behaviorReceptor agonistSignificant potentiationDependent ClLocomotor activityACh concentrationPainNociceptionReceptorsTonicG proteins
1987
Airway responses to nitrogen dioxide in asthmatic subjects
Mohsenin V. Airway responses to nitrogen dioxide in asthmatic subjects. Journal Of Toxicology And Environmental Health 1987, 22: 371-380. PMID: 3320381, DOI: 10.1080/15287398709531080.Peer-Reviewed Original ResearchConceptsAirway reactivityVital capacityAsthmatic subjectsDouble-blind randomized fashionPartial expiratory flowSpecific airway conductanceDose of methacholineNO2 exposureFunctional residual capacityAirway conductanceAirway responsesMethacholine inhalationExpiratory volumeLung functionExpiratory flowSignificant potentiationSignificant symptomsRandomized fashionRespiratory responsesResidual capacityAsthmaticsCommon indoor air pollutantsExposureSignificant changesDifferent days
1983
Potentiation of Insulin Action by a Sulfonylurea in Primary Cultures of Hepatocytes from Normal and Diabetic Rats
Salhanick A, Konowitz P, Amatruda J. Potentiation of Insulin Action by a Sulfonylurea in Primary Cultures of Hepatocytes from Normal and Diabetic Rats. Diabetes 1983, 32: 206-212. PMID: 6337899, DOI: 10.2337/diab.32.3.206.Peer-Reviewed Original ResearchConceptsDiabetic ratsInsulin actionInsulin responsivenessPrimary culturesStreptozotocin-diabetic ratsHepatic insulin resistanceDose-dependent increaseInsulin-dependent actionInsulin-stimulated ratesDependent diabetesDiabetic animalsInsulin resistanceNondiabetic animalsInsulin sensitivityAbsence of insulinInsulin secretionSignificant potentiationNormal ratsChronic exposureSpecific insulinRatsSerum-free mediumInsulinSulfonylurea tolazamideSulfonylureas
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