2025
Diuretic Potentiation Strategies in Acute Heart Failure
Siddiqi T, Packer M, Ezekowitz J, Fonarow G, Greene S, Kittleson M, Khan M, Mentz R, Testani J, Voors A, Butler J. Diuretic Potentiation Strategies in Acute Heart Failure. JACC Heart Failure 2025, 13: 14-27. PMID: 39779178, DOI: 10.1016/j.jchf.2024.09.017.Peer-Reviewed Original ResearchConceptsAcute heart failureHeart failureReceptor antagonistSodium-glucose cotransporter 2 inhibitorsLoop diuretic agentsMarkers of congestionMineralocorticoid receptor antagonistsVasopressin receptor antagonistsHeart failure eventsLong-term outcomesShort-term markersCarbonic anhydrase inhibitorsDiuretic strategyThiazide diureticsSerum creatinineDecongestion strategiesClinical outcomesConventional therapyDiuretic agentsImprove symptomsPhysical signsDiureticsCombination strategiesSymptomsAntagonist
2021
A Benzenesulfonamide-based Mitochondrial Uncoupler Induces Endoplasmic Reticulum Stress and Immunogenic Cell Death in Epithelial Ovarian Cancer
Bi F, Jiang Z, Park W, Hartwich TMP, Ge Z, Chong KY, Yang K, Morrison MJ, Kim D, Kim J, Zhang W, Kril LM, Watt DS, Liu C, Yang-Hartwich Y. A Benzenesulfonamide-based Mitochondrial Uncoupler Induces Endoplasmic Reticulum Stress and Immunogenic Cell Death in Epithelial Ovarian Cancer. Molecular Cancer Therapeutics 2021, 20: molcanther.mct-21-0396-a.2021. PMID: 34625503, PMCID: PMC8643344, DOI: 10.1158/1535-7163.mct-21-0396.Peer-Reviewed Original ResearchMeSH KeywordsAnimalsApoptosisCarbonic Anhydrase InhibitorsCarcinoma, Ovarian EpithelialCell Line, TumorEndoplasmic Reticulum StressFemaleHumansImmunogenic Cell DeathMiceMice, NudeSulfonamidesConceptsEpithelial ovarian cancerImmunogenic cell deathOvarian cancerTumor progressionAntitumor adaptive immune responsesDamage-associated molecular patternsCancer cellsMitochondrial uncouplerAdaptive immune responsesOvarian cancer modelCause of deathCurrent chemotherapeutic agentsNew therapeutic strategiesOvarian cancer cellsCancer cell proliferationCell deathEndoplasmic reticulum stressGynecologic malignanciesClinical outcomesEndoplasmic reticulum stress sensorNew anticancer therapiesPeritoneal fluidInduces Endoplasmic Reticulum StressImmune responseAbdominal cavity
1999
Characterization of ion transport mechanisms involved in bombesin-stimulated biliary secretion in rat cholangiocytes
Cho W, Boyer J. Characterization of ion transport mechanisms involved in bombesin-stimulated biliary secretion in rat cholangiocytes. Journal Of Hepatology 1999, 30: 1045-1051. PMID: 10406182, DOI: 10.1016/s0168-8278(99)80258-x.Peer-Reviewed Original ResearchMeSH Keywords4,4'-Diisothiocyanostilbene-2,2'-Disulfonic AcidAcetazolamideAnimalsBarium CompoundsBileBile DuctsBombesinCarbonic Anhydrase InhibitorsChloride ChannelsChloridesIn Vitro TechniquesIon TransportMaleMicroscopy, VideoNitrobenzoatesPotassium ChannelsRatsRats, Sprague-DawleyTetraethylammonium
1990
Treatment of humoral hypercalcemia of malignancy in rats with inhibitors of carbonic anhydrase
Brown G, Morris C, Mitnick M, Insogna K. Treatment of humoral hypercalcemia of malignancy in rats with inhibitors of carbonic anhydrase. Journal Of Bone And Mineral Research 1990, 5: 1037-1041. PMID: 1964358, DOI: 10.1002/jbmr.5650051007.Peer-Reviewed Original ResearchConceptsSerum calciumBone resorptionHumoral hypercalcemiaCarbonic anhydrase inhibitorsNephrogenous cyclic AMP excretionCyclic AMP excretionMean serum calciumOsteoclastic bone resorptionDrug-treated animalsLeydig cell tumorMechanism of actionUrine phosphorusUrine calciumSerum phosphorusCell tumorsAcetazolamide treatmentHypercalcemiaSignificant fallFisher ratsObserved hypercalcemiaResorptionDirect inhibitionSignificant riseMalignancyRats
1987
Carbonic Anhydrase Inhibitors
Preisig PA, Toto RD, Alpern RJ. Carbonic Anhydrase Inhibitors. 1987, 10: 136-159. PMID: 3133728, DOI: 10.1159/000173126.Peer-Reviewed Original ResearchMeSH KeywordsBicarbonatesBiological TransportCarbonic Anhydrase InhibitorsCarbonic AnhydrasesChloridesDiuresisHumansKidneyKidney Concentrating Ability
1973
Interaction of 13CO2 and Bicarbonate with Human Hemoglobin Preparations
Morrow J, Keim P, Visscher R, Marshall R, Gurd F. Interaction of 13CO2 and Bicarbonate with Human Hemoglobin Preparations. Proceedings Of The National Academy Of Sciences Of The United States Of America 1973, 70: 1414-1418. PMID: 4514311, PMCID: PMC433509, DOI: 10.1073/pnas.70.5.1414.Peer-Reviewed Original Research
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