Novel Approach to Performing Metabolite Identification in Drug Metabolism
Nassar A, Lee D. Novel Approach to Performing Metabolite Identification in Drug Metabolism. Journal Of Chromatographic Science 2007, 45: 113-119. PMID: 17462124, DOI: 10.1093/chromsci/45.3.113.Peer-Reviewed Original ResearchConceptsMetabolite identificationHuman liver microsomal incubationsMetabolite identification studiesDrug discoveryMS fragmentation patternsLiver microsomal incubationsLimit of detectionSite of metabolismDynamic-flow methodMass spectrometric analysisMultistage fragmentationMass spectrometerFragmentation patternsMicrosomal incubationsOnline separationChromatographic peaksMass spectrometryMinor metabolitesSpectrometric analysisFraction collectionO-dealkylationRadioactivity detectorMetabolite of dextromethorphanRadioactivity detectionColumn pressure
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