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Diacylglycerol Enhances Synaptic Vesicle Priming and Release

Publication Title: Roles for diacylglycerol in synaptic vesicle priming and release revealed by complete reconstitution of core protein machinery

Summary

Question
This study examined the molecular mechanisms underlying synaptic vesicle priming and release, focusing on the roles of diacylglycerol (DAG), Munc13, and Munc18 in facilitating neurotransmitter release. The researchers aimed to understand how these proteins interact to prepare synaptic vesicles for rapid calcium-triggered fusion.
Why it Matters
Neurotransmitter release is essential for communication between nerve cells, which underpins brain function and behavior. Understanding how synaptic vesicles are primed and released can provide insights into neurological processes and diseases, such as Alzheimer's and epilepsy, that involve disruptions in neurotransmitter signaling. This research could also inform the development of therapies targeting synaptic dysfunction.
Methods
The researchers used a biochemically defined in vitro system that reconstituted the core protein machinery involved in synaptic vesicle release. This included key proteins such as SNAREs (proteins essential for membrane fusion), Munc13, Munc18, Synaptotagmin, and Complexin. They tracked vesicle docking, priming, and calcium-triggered fusion using fluorescence microscopy and single-vesicle imaging techniques.
Key Findings
The study found that Munc18 acts as a nucleator for the SNARE complex, while Munc13 accelerates SNARE assembly in a DAG-dependent manner. Low concentrations of DAG improved vesicle priming and calcium-triggered release, while high concentrations reduced the regulatory 'clamping' mechanism, leading to spontaneous vesicle fusion. DAG binding to Munc13 significantly enhanced the formation of stably docked, release-ready vesicles and facilitated rapid fusion within milliseconds upon calcium influx.
Implications
These findings highlight the critical roles of Munc13, Munc18, and DAG in ensuring efficient neurotransmitter release. By elucidating how these proteins cooperate to prime synaptic vesicles, the research advances our understanding of synaptic function and its regulation. The results may have implications for treating neurological disorders characterized by impaired synaptic activity, offering potential targets for drug development.
Next Steps
The researchers suggest further studies to explore the structural transitions of Munc13 during vesicle priming and the molecular choreography of SNARE assembly. Additional research is needed to determine how DAG interacts with other regulatory elements in the synaptic vesicle fusion process.
Funding Information
This research was supported by the National Institutes of Health (NIH) under grants DK027044 and GM141194. The content is solely the responsibility of the authors and does not necessarily represent the official views of the National Institutes of Health. Yale University also provided funding and support for this research.
  • Proceedings of the National Academy of Sciences of the United States of America

    120 (34) - August 2023

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Full Citation

Sundaram R, Chatterjee A, Bera M, Grushin K, Panda A, Li F, Coleman J, Lee S, Ramakrishnan S, Ernst A, Gupta K, Rothman J, Krishnakumar S. Roles for diacylglycerol in synaptic vesicle priming and release revealed by complete reconstitution of core protein machinery. Proceedings Of The National Academy Of Sciences Of The United States Of America 2023, 120: e2309516120. PMID: 37590407, PMCID: PMC10450444, DOI: 10.1073/pnas.2309516120.
This AI-assisted summary has been reviewed and approved by at least one of the study's authors to ensure it accurately reflects the research.

Authors

  • Venkat Kalyana Sundaram, PhD

    First Author
    Yale School of Medicine

    Research Scientist in Cell Biology

  • Shyam Krishnakumar, PhD

    Last Author
    Yale School of Medicine

    Assistant Professor

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  • Proceedings of the National Academy of Sciences of the United States of America

    120 (34) - August 2023

    Read Full Publication
  • Engagement

    Citation
    Altmetric